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>an adenosine A1 receptor agonist elicits analgesia without cardiorespiratory depression” benzyloxy-cyclopentyladenosine (BnOCPA) >is an A1R selective agonist
by socky 4y ago
>an adenosine A1 receptor agonist elicits analgesia without cardiorespiratory depression”
benzyloxy-cyclopentyladenosine (BnOCPA)
>is an A1R selective agonist discovered to be a "potent and powerful analgesic,
but does not cause sedation, bradycardia, hypotension or respiratory depression"
https://en.m.wikipedia.org/wiki/Adenosine_A1_receptor https://en.m.wikipedia.org/wiki/Adenosine_A1_receptor
Selective activation of Gαob by an adenosine A1 receptor agonist elicits analgesia without cardiorespiratory depression
https://www.nature.com/articles/s41467-022-31652-2 https://www.nature.com/articles/s41467-022-31652-2